Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50016430
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594943(CHEMBL5172462)
Affinity DataKd:  2.71E+3nMAssay Description:Binding affinity to biotinylated EED (unknown origin) assessed as dissociation constant incubated for 120 secsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594939(CHEMBL5187105)
Affinity DataKd:  900nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594940(CHEMBL5174215)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594941(CHEMBL5191512)
Affinity DataKd:  5.20E+3nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594942(CHEMBL5204429)
Affinity DataKd:  163nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM291687(US9580437, Example 2 | N-((5-Fluoro-2,3-dihydroben...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50563656(CHEMBL4754048)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50563657(CHEMBL4762963)
Affinity DataKd:  2.40nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50563659(CHEMBL4759335)
Affinity DataKd:  0.5nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50563658(CHEMBL4748924)
Affinity DataKd:  15nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50282163(CHEMBL4171889)
Affinity DataKd:  680nMAssay Description:Binding affinity to N-terminal His-tagged full length EED (unknown origin) by ITC methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50282157(CHEMBL4161291)
Affinity DataKd:  1.14E+3nMAssay Description:Binding affinity to N-terminal His-tagged full length EED (unknown origin) by ITC methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50282164(CHEMBL4164708)
Affinity DataKd:  8.82E+3nMAssay Description:Binding affinity to N-terminal His-tagged full length EED (unknown origin) by ITC methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50096619(CHEMBL97453 | 1,8,9-Trihydroxy-3-methoxy-benzo[4,5...)
Affinity DataKd:  2.82E+3nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant SPR assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKd:  1.51E+4nMAssay Description:Binding affinity to EED (unknown origin) assessed as dissociation constant SPR assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594945(CHEMBL5180485)
Affinity DataKd:  0.631nMAssay Description:Binding affinity to human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50562610(CHEMBL4779022)
Affinity DataKd:  0.537nMAssay Description:Binding affinity to human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594938(CHEMBL5201204)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of His-tagged EED (unknown origin) incubated for 30 mins in presence of biotinylated H3K27me3 peptide (19 to 33 aa) by alpha screening com...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594938(CHEMBL5201204)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM291687(US9580437, Example 2 | N-((5-Fluoro-2,3-dihydroben...)
Affinity DataIC50: 5nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594945(CHEMBL5180485)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50562610(CHEMBL4779022)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHistone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594944(CHEMBL5181703)
Affinity DataIC50: 18nMAssay Description:Inhibition of PRC2 complex of EZH2-EED-SUZ12 (unknown origin) using human nucleosome as substrate incubated for 70 mins in presence of [3H]SAMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594928(CHEMBL5171195)
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM225230(EED226 | US11013745, Compound EED226)
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594929(CHEMBL5173010)
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594931(CHEMBL5169768)
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594930(CHEMBL5188142)
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM225230(EED226 | US11013745, Compound EED226)
Affinity DataIC50: 45nMAssay Description:Inhibition of full length N-terminal His-6x tagged EED (1 to 441 residues) (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM291687(US9580437, Example 2 | N-((5-Fluoro-2,3-dihydroben...)
Affinity DataIC50: 60nMAssay Description:Inhibition of EED (unknown origin) by alpha screen binding assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594937(CHEMBL5180270)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594932(CHEMBL5203240)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594933(CHEMBL5193972)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594934(CHEMBL5171965)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594935(CHEMBL5205261)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594936(CHEMBL5206890)
Affinity DataIC50: 100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50562612(CHEMBL4749741)
Affinity DataIC50: 247nMAssay Description:Inhibition of full length N-terminal His-6x tagged EED (1 to 441 residues) (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM223986((3R,4S)-1-[(1S)-7-fluoroindan-1-yl]-N,N-dimethyl-4...)
Affinity DataIC50: 290nMAssay Description:Inhibition of GST-tagged EED in human G-401 cells assessed as inhibition of histone trimethylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50562612(CHEMBL4749741)
Affinity DataIC50: 300nMAssay Description:Inhibition of EZH2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50236003(CHEMBL4096234)
Affinity DataIC50: 620nMAssay Description:Inhibition of biotinylated H3K27Me3 peptide (19 to 33 aa) binding to EED (1 to 441 residues) (unknown origin) expressed in Escherichia coli BL21-Codo...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50235994(CHEMBL4063655)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594939(CHEMBL5187105)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594941(CHEMBL5191512)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50236003(CHEMBL4096234)
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of EED in human G-401 cells assessed as reduction of global H3K27Me3 level by ELISAMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50236003(CHEMBL4096234)
Affinity DataIC50: 4.03E+3nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594940(CHEMBL5174215)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM225230(EED226 | US11013745, Compound EED226)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50594944(CHEMBL5181703)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to GST-tagged EED (unknown origin) assessed as inhibition constant incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPolycomb protein EED(Human)
Sanquan College of Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM223986((3R,4S)-1-[(1S)-7-fluoroindan-1-yl]-N,N-dimethyl-4...)
Affinity DataKi:  11nMAssay Description:Binding affinity to GST-tagged EED (unknown origin) assessed as inhibition constant incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)