Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50017570
TargetBromodomain testis-specific protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  1.12E+3nMAssay Description:Binding affinity to His6-tagged human BRDT bromodomain-1 (21 to 137 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  360nMAssay Description:Binding affinity to His6-tagged human BRD4 bromodomain-1 (44 to 168 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602884(CHEMBL5179520)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to His6-tagged human BRD3 bromodomain-2 (306 to 416 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  1.51E+3nMAssay Description:Binding affinity to His6-tagged human BRD3 bromodomain-2 (306 to 416 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  560nMAssay Description:Binding affinity to His6-tagged human BRD3 bromodomain-1 (24 to 144 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602884(CHEMBL5179520)
Affinity DataKd:  840nMAssay Description:Binding affinity to His6-tagged human BRD2 bromodomain-1 (77 to 194 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  390nMAssay Description:Binding affinity to His6-tagged human BRD2 bromodomain-1 (77 to 194 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 9(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  2.61E+3nMAssay Description:Binding affinity to His6-tagged human BRD9 bromodomain (14 to 134 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602884(CHEMBL5179520)
Affinity DataKd:  58nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602873(CHEMBL5191045)
Affinity DataKd:  36nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602870(CHEMBL5192405)
Affinity DataKd:  44nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602865(CHEMBL5205974)
Affinity DataKd:  30nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50311385(CHEMBL4171749)
Affinity DataKd:  165nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataKd:  14nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50178219(CHEMBL3814752)
Affinity DataKd:  68nMAssay Description:Binding affinity to His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation const...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602881(CHEMBL5204688)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602873(CHEMBL5191045)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602864(INOBRODIB | Inobrodib | Ccs 1477 | Ccs1477 | CCS-1...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602874(CHEMBL5179328)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602878(CHEMBL5179809)
Affinity DataIC50: 3nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602884(CHEMBL5179520)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602865(CHEMBL5205974)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602869(CHEMBL5198394)
Affinity DataIC50: 12nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602868(CHEMBL5195756)
Affinity DataIC50: 13nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602871(CHEMBL5191527)
Affinity DataIC50: 14nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50178219(CHEMBL3814752)
Affinity DataIC50: 14nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602880(CHEMBL5192803)
Affinity DataIC50: 21nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602872(CHEMBL5195875)
Affinity DataIC50: 22nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602879(CHEMBL5198835)
Affinity DataIC50: 25nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602870(CHEMBL5192405)
Affinity DataIC50: 26nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602883(CHEMBL5208356)
Affinity DataIC50: 26nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602876(CHEMBL5200678)
Affinity DataIC50: 42nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602867(CHEMBL5207470)
Affinity DataIC50: 55nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602875(CHEMBL5204233)
Affinity DataIC50: 56nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602866(CHEMBL5179738)
Affinity DataIC50: 70nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602877(CHEMBL5181127)
Affinity DataIC50: 78nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50602882(CHEMBL5192554)
Affinity DataIC50: 79nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCREB-binding protein(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50311385(CHEMBL4171749)
Affinity DataIC50: 178nMAssay Description:Inhibition of His6-tagged human CBP bromodomain (1081 to 1197 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed