Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50016632
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596260(CHEMBL5183506)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataEC50:  2.50E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596277(CHEMBL5198009)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596276(CHEMBL5207002)
Affinity DataEC50:  7.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596275(CHEMBL5176348)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596274(CHEMBL5204986)
Affinity DataEC50:  8.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596273(CHEMBL5185133)
Affinity DataEC50:  2.50E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596272(CHEMBL5199813)
Affinity DataEC50:  3.80E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596271(CHEMBL5176046)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596270(CHEMBL5186572)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596269(CHEMBL5183842)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596268(CHEMBL5203592)
Affinity DataEC50:  500nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596267(CHEMBL5172698)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596266(CHEMBL5205450)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596265(CHEMBL5178897)
Affinity DataEC50:  2.60E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596264(CHEMBL5206355)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596263(CHEMBL5207657)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596262(CHEMBL5176331)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596272(CHEMBL5199813)
Affinity DataIC50: 190nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 230nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596263(CHEMBL5207657)
Affinity DataIC50: 280nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataIC50: 280nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataIC50: 340nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataIC50: 370nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596275(CHEMBL5176348)
Affinity DataIC50: 370nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596271(CHEMBL5176046)
Affinity DataIC50: 460nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596264(CHEMBL5206355)
Affinity DataIC50: 480nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596274(CHEMBL5204986)
Affinity DataIC50: 540nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596262(CHEMBL5176331)
Affinity DataIC50: 680nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596262(CHEMBL5176331)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596264(CHEMBL5206355)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596272(CHEMBL5199813)
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596275(CHEMBL5176348)
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 3.84E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataIC50: 6.46E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataIC50: 7.64E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 9.16E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596263(CHEMBL5207657)
Affinity DataIC50: 9.92E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596271(CHEMBL5176046)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596274(CHEMBL5204986)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based microtiter plate ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596269(CHEMBL5183842)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596269(CHEMBL5183842)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In DepthDetails
PubMed