Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50014967
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581594(CHEMBL5086897)
Affinity DataKd:  200nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581601(CHEMBL5079045)
Affinity DataKd:  143nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581600(CHEMBL5086339)
Affinity DataKd:  236nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581599(CHEMBL5087181)
Affinity DataKd:  63nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581598(CHEMBL5081695)
Affinity DataKd:  246nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581597(CHEMBL5074720)
Affinity DataKd:  66nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581596(CHEMBL5075400)
Affinity DataKd:  98nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581595(CHEMBL4215078)
Affinity DataKd:  34nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50459880(CHEMBL4226570)
Affinity DataKd:  34nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581587(CHEMBL5087145)
Affinity DataKd:  119nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581593(CHEMBL5086047)
Affinity DataKd:  200nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581592(CHEMBL5094871)
Affinity DataKd:  170nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581591(CHEMBL5087530)
Affinity DataKd:  170nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50099062(CHEMBL3344081 | US10730870, Example 3 | US11512083...)
Affinity DataKd:  113nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581590(CHEMBL5081396)
Affinity DataKd:  144nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581589(CHEMBL4793272)
Affinity DataKd:  138nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50581588(CHEMBL5082521)
Affinity DataKd:  136nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues) (unknown origin) expressed in Escherichia coli assessed as displacement of HIF-1a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed