Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50017542
TargetCasein kinase I isoform alpha-like(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to CK1a1L (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform epsilon(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKd:  100nMAssay Description:Binding affinity to CK1epsilon (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of P38alphaMAPK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetMitogen-activated protein kinase 11(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of P38betaMAPK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(trans -1-(4-hydroxycyclohexyl)-4-(4-fluorophenyl)-...)
Affinity DataIC50: 44nMAssay Description:Inhibition of P38alphaMAPK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetMitogen-activated protein kinase 11(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(trans -1-(4-hydroxycyclohexyl)-4-(4-fluorophenyl)-...)
Affinity DataIC50: 44nMAssay Description:Inhibition of P38betaMAPK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50602625(CHEMBL5172162)
Affinity DataIC50: 70nMAssay Description:Inhibition of c-Raf (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(trans -1-(4-hydroxycyclohexyl)-4-(4-fluorophenyl)-...)
Affinity DataKi:  25nMAssay Description:Binding affinity to CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform delta(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKi:  39nMAssay Description:Binding affinity to CK1delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(trans -1-(4-hydroxycyclohexyl)-4-(4-fluorophenyl)-...)
Affinity DataKi:  501nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
Christian-Albrechts University of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKi:  650nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed