Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50018429
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50161957(CHEMBL180022 | N-(4-(3-chloro-4-(pyridin-2-ylmetho...)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant HER4 (unknown origin) expressed in baculovirus infected sf9 cells autophosphorylation incubated for 1 hrs in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50161957(CHEMBL180022 | N-(4-(3-chloro-4-(pyridin-2-ylmetho...)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant HER2 (676 to 1255 residues) (unknown origin) expressed in baculovirus infected sf9 cells autophosphorylation incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50161957(CHEMBL180022 | N-(4-(3-chloro-4-(pyridin-2-ylmetho...)
Affinity DataIC50: 92nMAssay Description:Inhibition of recombinant HER1 (645 to 1186 residues) (unknown origin) expressed in baculovirus infected sf9 cells autophosphorylation incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed