Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50014166
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to 5FW-labeled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by BODIPY-BI2536 tracer ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  230nMAssay Description:Binding affinity to BRD9 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  0.240nMAssay Description:Binding affinity to BRD9 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  0.470nMAssay Description:Binding affinity to BRD9 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 7(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  0.760nMAssay Description:Binding affinity to BRD7 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  11nMAssay Description:Binding affinity to CECR2 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  44nMAssay Description:Binding affinity to GCN5L2 (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataKd:  300nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  370nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  14nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  12nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  70nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  6.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to 5FW-labeled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by BODIPY-BI2536 tracer ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataIC50: 36nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataIC50: 56nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataIC50: 67nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573198(CHEMBL4848138)
Affinity DataIC50: 170nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50234940(CHEMBL4101756)
Affinity DataIC50: 220nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573192(CHEMBL4850516)
Affinity DataIC50: 250nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573190(CHEMBL4866748)
Affinity DataIC50: 290nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573191(CHEMBL4870218)
Affinity DataIC50: 310nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573193(CHEMBL4848082)
Affinity DataIC50: 370nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataIC50: 380nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573202(CHEMBL4877696)
Affinity DataIC50: 550nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573188(CHEMBL4850913)
Affinity DataIC50: 700nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573204(CHEMBL4863529)
Affinity DataIC50: 790nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573195(CHEMBL4855881)
Affinity DataIC50: 800nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50234924(CHEMBL4065579)
Affinity DataIC50: 950nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573196(CHEMBL4877118)
Affinity DataIC50: 970nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50234923(CHEMBL4069412)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573187(CHEMBL4861822)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573194(CHEMBL4858548)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573186(CHEMBL4872107)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573185(CHEMBL4853420)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573199(CHEMBL4849136)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573183(CHEMBL4867912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573189(CHEMBL4857332)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50234944(CHEMBL4072538 | US10239861, Example 60)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of HIS9-tagged BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573184(CHEMBL4871852)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573202(CHEMBL4877696)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIS9-tagged BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573190(CHEMBL4866748)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of HIS9-tagged BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of HIS9-tagged BRD4 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed