Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50014698
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579208(CHEMBL4867107)
Affinity DataIC50: 2nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579222(CHEMBL4861383)
Affinity DataIC50: 2.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518526(US11124518, Example 1 | 2-Allyl-1-(6-(2-hydroxypro...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518531(US11124518, Example 6 | 2-Allyl-1-(6-(2-hydroxypro...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518527(US11124518, Example 2 | 2-Alyl-6-((2′,3̸...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518538(US11124518, Example 13 | 2-Allyl-6-((2-(2-hydroxye...)
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579228(CHEMBL4867211)
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518530(US11124518, Example 5 | 2-Allyl-1-(6-(2-hydroxypro...)
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM518540(US11124518, Example 16 | 2-Allyl-1-(6-(2-hydroxypr...)
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579225(CHEMBL4874546)
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579214(CHEMBL4856035)
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579218(CHEMBL4876612)
Affinity DataIC50: 2.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579223(CHEMBL4853285)
Affinity DataIC50: 3.10nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579224(CHEMBL4861351)
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579227(CHEMBL4847705)
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579221(CHEMBL4866800)
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579216(CHEMBL4865963)
Affinity DataIC50: 3.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579213(CHEMBL4853973)
Affinity DataIC50: 3.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579220(CHEMBL4868683)
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579219(CHEMBL4857841)
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579215(CHEMBL4861168)
Affinity DataIC50: 4.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579211(CHEMBL4871803)
Affinity DataIC50: 4.80nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579212(CHEMBL4879157)
Affinity DataIC50: 5.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579210(CHEMBL4853185)
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579210(CHEMBL4853185)
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579209(CHEMBL4874090)
Affinity DataIC50: 6.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579226(CHEMBL4856253)
Affinity DataIC50: 12nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579229(CHEMBL4863657)
Affinity DataIC50: 22nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 40nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 19(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 59nMAssay Description:Inhibition of YSK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 60nMAssay Description:Inhibition of EGFR d747-749/A750P mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579231(CHEMBL4847051)
Affinity DataIC50: 64nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 70nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetWee1-like protein kinase(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579230(CHEMBL4877772)
Affinity DataIC50: 100nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 227nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579208(CHEMBL4867107)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Zentalis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50579217(CHEMBL4871593)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed