Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50014535
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM418817(US10450297, Example 317 | US10450297, Example 318 ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of JAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of TYK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fes/Fps(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of Fes (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577163(CHEMBL4851157)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of Fyn (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of Lck (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577167(CHEMBL4873104)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577176(CHEMBL4846553)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577188(CHEMBL4874196)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577187(CHEMBL4853724)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577177(CHEMBL4854620)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577168(CHEMBL4877875)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577171(CHEMBL4857298)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 14nMAssay Description:Inhibition of CK2alpha1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577160(CHEMBL4846093)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577170(CHEMBL4872520)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577165(CHEMBL4878656)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577182(CHEMBL4849384)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577154(CHEMBL4861088)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577180(CHEMBL4861397)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577189(CHEMBL4862392)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 22nMAssay Description:Inhibition of ROS (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577155(CHEMBL4858365)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577192(CHEMBL4860735)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetEphrin type-B receptor 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 30nMAssay Description:Inhibition of EphB1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577164(CHEMBL4871809)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577178(CHEMBL4867151)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577190(CHEMBL4867910)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577161(CHEMBL4877120)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577186(CHEMBL4861021)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577156(CHEMBL4876873)
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577193(CHEMBL4876098)
Affinity DataIC50: 54nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577157(CHEMBL4879263)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577185(CHEMBL4873271)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577166(CHEMBL4874015)
Affinity DataIC50: 68nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577162(CHEMBL4869934)
Affinity DataIC50: 78nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577159(CHEMBL4874892)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577191(CHEMBL4879025)
Affinity DataIC50: 126nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577181(CHEMBL4878892)
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577184(CHEMBL4867693)
Affinity DataIC50: 321nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Yonsei University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50577179(CHEMBL4849868)
Affinity DataIC50: 361nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
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