Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50015509
TargetHeat shock protein HSP 90-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  8.20E+3nMAssay Description:Binding affinity to Hsp90alpha (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataKon:  0.0284M-1s-1Assay Description:Binding affinity to GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant at 0.37 to 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataKon:  0.114M-1s-1Assay Description:Binding affinity to His-tagged human N-terminal HSP90alpha (1 to 236 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587146(CHEMBL5073759)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataKd:  220nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataKd:  200nMAssay Description:Binding affinity to Grp94 (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataKd: >2.50E+5nMAssay Description:Binding affinity to Hsp90alpha (unknown origin) by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50005782(ATI-13387X | ONALESPIB)
Affinity DataIC50: 13nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50450705(CHEMBL4170630)
Affinity DataIC50: 20nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587115(CHEMBL5093243)
Affinity DataIC50: 60nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587119(CHEMBL5089044)
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587134(CHEMBL5079918)
Affinity DataIC50: 203nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587116(CHEMBL5084235)
Affinity DataIC50: 205nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587120(CHEMBL5090316)
Affinity DataIC50: 210nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587132(CHEMBL5089381)
Affinity DataIC50: 234nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587118(CHEMBL5084137)
Affinity DataIC50: 251nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587130(CHEMBL5094079)
Affinity DataIC50: 310nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587114(CHEMBL5087678)
Affinity DataIC50: 313nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587113(CHEMBL5093787)
Affinity DataIC50: 325nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587133(CHEMBL5090818)
Affinity DataIC50: 393nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587117(CHEMBL5087889)
Affinity DataIC50: 519nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587138(CHEMBL5084856)
Affinity DataIC50: 528nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587137(CHEMBL5087347)
Affinity DataIC50: 627nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587139(CHEMBL5091405)
Affinity DataIC50: 797nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587112(CHEMBL5075059)
Affinity DataIC50: 914nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587131(CHEMBL5077310)
Affinity DataIC50: 947nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587142(CHEMBL5090524)
Affinity DataIC50: 985nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587140(CHEMBL5070758)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587141(CHEMBL5093202)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587135(CHEMBL5088257)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587129(CHEMBL5087473)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587145(CHEMBL5092629)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587127(CHEMBL5089184)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587144(CHEMBL5075220)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587126(CHEMBL5081112)
Affinity DataIC50: 2.77E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587128(CHEMBL5089014)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587143(CHEMBL5077569)
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587123(CHEMBL5076003)
Affinity DataIC50: 6.84E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587125(CHEMBL5082207)
Affinity DataIC50: 7.54E+3nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587124(CHEMBL5085266)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587136(CHEMBL5088079)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587121(CHEMBL5091953)
Affinity DataIC50: 6.26E+4nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50587122(CHEMBL5092143)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed