Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 50014743
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579684(CHEMBL5083054)
Affinity DataEC50:  372nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579694(CHEMBL5075230)
Affinity DataEC50:  237nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579693(CHEMBL5092182)
Affinity DataEC50:  166nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579692(CHEMBL5086009)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579691(CHEMBL5087233)
Affinity DataEC50:  578nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579690(CHEMBL5075508)
Affinity DataEC50:  619nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579689(CHEMBL5084909)
Affinity DataEC50:  683nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579688(CHEMBL5080082)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579687(CHEMBL5075266)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579686(CHEMBL5085975)
Affinity DataEC50:  376nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579685(CHEMBL5093957)
Affinity DataEC50:  259nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579695(CHEMBL5081645)
Affinity DataEC50:  354nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579683(CHEMBL5092277)
Affinity DataEC50:  406nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50121214(CHEMBL3623075)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579682(CHEMBL5085472)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579681(CHEMBL5079935)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579680(CHEMBL5088300)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579679(CHEMBL5078948)
Affinity DataEC50:  4.15E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579678(CHEMBL5089837)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579677(CHEMBL5088669)
Affinity DataEC50:  2.13E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579676(CHEMBL5086127)
Affinity DataEC50:  560nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579675(CHEMBL5089335)
Affinity DataEC50:  753nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579706(CHEMBL5080486)
Affinity DataEC50:  99nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579711(CHEMBL5091326)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human OX2R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM514588(US11098029, Example 24)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human OX2R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM386067(methyl (2R,3S)-3- ((methylsulfonyl)amino)-2-(((cis...)
Affinity DataEC50:  5.50E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579710(CHEMBL1198149)
Affinity DataEC50: >3.20E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579711(CHEMBL5091326)
Affinity DataEC50: >3.55E+4nMAssay Description:Agonist activity at human OX1R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM386067(methyl (2R,3S)-3- ((methylsulfonyl)amino)-2-(((cis...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human OX1R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579710(CHEMBL1198149)
Affinity DataEC50: >3.20E+3nMAssay Description:Agonist activity at human OX1R stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579709(CHEMBL5087440)
Affinity DataEC50:  863nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579708(CHEMBL3623078)
Affinity DataEC50:  1.27E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579707(CHEMBL5087774)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579674(CHEMBL5082761)
Affinity DataEC50:  252nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579705(CHEMBL5070320)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579704(CHEMBL5094915)
Affinity DataEC50:  134nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579703(CHEMBL5083235)
Affinity DataEC50:  464nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579702(CHEMBL5084798)
Affinity DataEC50:  107nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579701(CHEMBL5084458)
Affinity DataEC50:  532nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579700(CHEMBL5090790)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579699(CHEMBL5091029)
Affinity DataEC50:  1.63E+3nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579698(CHEMBL5082069)
Affinity DataEC50:  293nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579697(CHEMBL5079739)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579696(CHEMBL5086661)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX2R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579682(CHEMBL5085472)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579691(CHEMBL5087233)
Affinity DataEC50:  5.17E+3nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579690(CHEMBL5075508)
Affinity DataEC50:  7.53E+3nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579689(CHEMBL5084909)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579688(CHEMBL5080082)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50579687(CHEMBL5075266)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
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