Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50012468
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557812(CHEMBL4786074)
Affinity DataIC50: 6nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557813(CHEMBL4763312)
Affinity DataIC50: 9nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557832(CHEMBL4742368)
Affinity DataIC50: 10nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50200880(2-hydroxy-N,N-dimethyl-3-{2-[[(R)-1-(5-methylfuran...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557814(CHEMBL4757674)
Affinity DataIC50: 15nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557830(CHEMBL4746698)
Affinity DataIC50: 29nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557826(CHEMBL4747035)
Affinity DataIC50: 43nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557821(CHEMBL4752486)
Affinity DataIC50: 54nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557825(CHEMBL4793352)
Affinity DataIC50: 68nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557834(CHEMBL4741864)
Affinity DataIC50: 98nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557824(CHEMBL4750465)
Affinity DataIC50: 140nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50200880(2-hydroxy-N,N-dimethyl-3-{2-[[(R)-1-(5-methylfuran...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557823(CHEMBL4800297)
Affinity DataIC50: 269nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557820(CHEMBL4799848)
Affinity DataIC50: 305nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557827(CHEMBL4746803)
Affinity DataIC50: 305nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557828(CHEMBL4786309)
Affinity DataIC50: 470nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557819(CHEMBL4757462)
Affinity DataIC50: 915nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557822(CHEMBL4797191)
Affinity DataIC50: 2.19E+3nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557831(CHEMBL4755486)
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557829(CHEMBL4762597)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557833(CHEMBL4745933)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557812(CHEMBL4786074)
Affinity DataIC50: 4.70E+3nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557813(CHEMBL4763312)
Affinity DataIC50: 5.40E+3nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557832(CHEMBL4742368)
Affinity DataIC50: 9.10E+3nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557825(CHEMBL4793352)
Affinity DataIC50: 1.47E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50506089(CHEMBL4536494)
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557830(CHEMBL4746698)
Affinity DataIC50: 2.03E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557821(CHEMBL4752486)
Affinity DataIC50: 2.17E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557814(CHEMBL4757674)
Affinity DataIC50: 2.34E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557817(CHEMBL4777637)
Affinity DataIC50: 2.36E+4nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557835(CHEMBL4760919)
Affinity DataIC50: 2.50E+4nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557818(CHEMBL4765070)
Affinity DataIC50: 2.97E+4nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557819(CHEMBL4757462)
Affinity DataIC50: 3.81E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557827(CHEMBL4746803)
Affinity DataIC50: 4.18E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557820(CHEMBL4799848)
Affinity DataIC50: 4.78E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557832(CHEMBL4742368)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557826(CHEMBL4747035)
Affinity DataIC50: 5.46E+4nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557818(CHEMBL4765070)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557822(CHEMBL4797191)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557823(CHEMBL4800297)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557824(CHEMBL4750465)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557815(CHEMBL4781979)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557817(CHEMBL4777637)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557828(CHEMBL4786309)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557829(CHEMBL4762597)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557816(CHEMBL4797342)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557831(CHEMBL4755486)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557815(CHEMBL4781979)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557833(CHEMBL4745933)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50557834(CHEMBL4741864)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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