Compile Data Set for Download or QSAR
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 50013947
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50564412(CHEMBL4800654)
Affinity DataEC50:  120nMAssay Description:Agonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571106(CHEMBL4853580)
Affinity DataEC50:  120nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571107(CHEMBL4853571)
Affinity DataEC50:  5.44E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571108(CHEMBL4870760)
Affinity DataEC50:  1.01E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571110(CHEMBL4851237)
Affinity DataEC50:  1.01E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571111(CHEMBL4851145)
Affinity DataEC50:  1.89E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataEC50:  3.80E+4nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571114(CHEMBL4871032)
Affinity DataEC50:  6.51E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571115(CHEMBL4849503)
Affinity DataEC50:  415nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571118(CHEMBL4861959)
Affinity DataEC50:  180nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571119(CHEMBL4852827)
Affinity DataEC50:  128nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571120(CHEMBL4862515)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571123(CHEMBL4869951)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571125(CHEMBL4875988)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571126(CHEMBL4859208)
Affinity DataEC50:  6.12E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571127(CHEMBL4855745)
Affinity DataEC50:  4.62E+3nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571128(CHEMBL4869562)
Affinity DataEC50:  122nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571129(CHEMBL4862733)
Affinity DataEC50:  102nMAssay Description:Agonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as transcriptional activities by measuring ERE driven reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant HDAC8 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant HDAC6 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50564412(CHEMBL4800654)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571125(CHEMBL4875988)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571124(CHEMBL4874242)
Affinity DataIC50: 114nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571116(CHEMBL4874175)
Affinity DataIC50: 129nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571109(CHEMBL4855191)
Affinity DataIC50: 146nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50564412(CHEMBL4800654)
Affinity DataIC50: 633nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571119(CHEMBL4852827)
Affinity DataIC50: 1.11E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571121(CHEMBL4870293)
Affinity DataIC50: 1.17E+3nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571107(CHEMBL4853571)
Affinity DataIC50: 1.25E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571114(CHEMBL4871032)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human recombinant HDAC6 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571111(CHEMBL4851145)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571130(CHEMBL4849015)
Affinity DataIC50: 1.45E+3nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571123(CHEMBL4869951)
Affinity DataIC50: 1.87E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571113(CHEMBL4868001)
Affinity DataIC50: 1.88E+3nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571116(CHEMBL4874175)
Affinity DataIC50: 2.08E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataIC50: 2.11E+3nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571130(CHEMBL4849015)
Affinity DataIC50: 2.32E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571122(CHEMBL4878251)
Affinity DataIC50: 2.61E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571121(CHEMBL4870293)
Affinity DataIC50: 3.13E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of human recombinant HDAC8 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571117(CHEMBL4873312)
Affinity DataIC50: 3.68E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571114(CHEMBL4871032)
Affinity DataIC50: 3.94E+3nMAssay Description:Inhibition of human recombinant HDAC8 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataIC50: 4.53E+3nMAssay Description:Inhibition of human recombinant HDAC6 incubated for 15 mins by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571112(CHEMBL4855392)
Affinity DataIC50: 5.08E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571113(CHEMBL4868001)
Affinity DataIC50: 5.27E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571115(CHEMBL4849503)
Affinity DataIC50: 5.67E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571110(CHEMBL4851237)
Affinity DataIC50: 5.78E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571124(CHEMBL4874242)
Affinity DataIC50: 5.90E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571126(CHEMBL4859208)
Affinity DataIC50: 6.12E+3nMAssay Description:Antagonist activity at ERalpha (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50571122(CHEMBL4878251)
Affinity DataIC50: 7.09E+3nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human HEK293T cells assessed as inhibition of 17beta-estradiol-induced transcriptional ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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