Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50014855
TargetGABA A receptor alpha-4/beta-3/gamma-2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 1.00E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha4beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGABA A receptor alpha-1/beta-1/gamma-2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 1.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta1gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 5.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha3beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 1.57E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha2beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 1.94E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha5beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50: 2.10E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed