Compile Data Set for Download or QSAR
Report error Found 135 Enz. Inhib. hit(s) with all data for entry = 50014651
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataEC50:  1.01E+3nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human recombinant CB1 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataEC50:  188nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578445(CHEMBL4852456)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578456(CHEMBL4846991)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO-K1 cell membrane assessed as increase in GTPgammaS binding pretreated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578464(CHEMBL4863350)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578464(CHEMBL4863350)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578456(CHEMBL4846991)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578456(CHEMBL4846991)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578454(CHEMBL4854325)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578454(CHEMBL4854325)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578460(CHEMBL4857976)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578460(CHEMBL4857976)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578434(CHEMBL4877653)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578434(CHEMBL4877653)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578452(CHEMBL4850004)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578452(CHEMBL4850004)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578445(CHEMBL4852456)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578445(CHEMBL4852456)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578432(CHEMBL4862930)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578458(CHEMBL4849400)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578458(CHEMBL4849400)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578462(CHEMBL4847976)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578434(CHEMBL4877653)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578434(CHEMBL4877653)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578427(CHEMBL4852553)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578427(CHEMBL4852553)
Affinity DataKi:  196nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50398220(CHEMBL2181540)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578425(CHEMBL4850969)
Affinity DataKi:  217nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578425(CHEMBL4850969)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578429(CHEMBL4852077)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578429(CHEMBL4852077)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578427(CHEMBL4852553)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578427(CHEMBL4852553)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50398220(CHEMBL2181540)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578441(CHEMBL4865342)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578441(CHEMBL4865342)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50398222(CHEMBL2177264)
Affinity DataKi:  465nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578423(CHEMBL4862523)
Affinity DataKi:  486nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578423(CHEMBL4862523)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Karlsruhe Institute of Technology (Kit)

Curated by ChEMBL
LigandPNGBDBM50578424(CHEMBL4860325)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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