Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50013478
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 0.430nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 0.530nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566467(CHEMBL4867132)
Affinity DataIC50: 6.90nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566445(CHEMBL4852725)
Affinity DataIC50: 8.10nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 9nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566464(CHEMBL4849980)
Affinity DataIC50: 12nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566446(CHEMBL4866685)
Affinity DataIC50: 13nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566468(CHEMBL4853767)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566447(CHEMBL4865371)
Affinity DataIC50: 13nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50098563(Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 14nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566467(CHEMBL4867132)
Affinity DataIC50: 14nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566468(CHEMBL4853767)
Affinity DataIC50: 16nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566454(CHEMBL4861024)
Affinity DataIC50: 36nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566452(CHEMBL4848344)
Affinity DataIC50: 36nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566453(CHEMBL4865509)
Affinity DataIC50: 37nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566448(CHEMBL4857992)
Affinity DataIC50: 37nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566461(CHEMBL4869368)
Affinity DataIC50: 37nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566463(CHEMBL4876499)
Affinity DataIC50: 37nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566464(CHEMBL4849980)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566462(CHEMBL4875003)
Affinity DataIC50: 44nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566465(CHEMBL4870505)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human GIPR expressed in HEK293 cells assessed as inhibition of GIP-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566457(CHEMBL4876838)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566453(CHEMBL4865509)
Affinity DataIC50: 73nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566454(CHEMBL4861024)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566466(CHEMBL4870133)
Affinity DataIC50: 81nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566458(CHEMBL4860642)
Affinity DataIC50: 82nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566462(CHEMBL4875003)
Affinity DataIC50: 95nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human GLP-1R expressed in HEK293 cells assessed as inhibition of GLP1-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566457(CHEMBL4876838)
Affinity DataIC50: 107nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566465(CHEMBL4870505)
Affinity DataIC50: 114nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGastric inhibitory polypeptide receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 125nMAssay Description:Antagonist activity at mouse GIPR expressed in CHO-K1 cells assessed as inhibition of GIP-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566463(CHEMBL4876499)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 131nMAssay Description:Antagonist activity at mouse GLP1R expressed in CHO-K1 cells assessed as inhibition of GLP1-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566451(CHEMBL4875380)
Affinity DataIC50: 136nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566458(CHEMBL4860642)
Affinity DataIC50: 146nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566456(CHEMBL4876913)
Affinity DataIC50: 163nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566461(CHEMBL4869368)
Affinity DataIC50: 192nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566466(CHEMBL4870133)
Affinity DataIC50: 267nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566451(CHEMBL4875380)
Affinity DataIC50: 275nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566459(CHEMBL4850520)
Affinity DataIC50: 346nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566460(CHEMBL4873721)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566456(CHEMBL4876913)
Affinity DataIC50: 472nMAssay Description:Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566449(CHEMBL4846293)
Affinity DataIC50: 983nMAssay Description:Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GIPR expressed in HEK293 cells assessed as inhibition of GIP-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GLP-1R expressed in HEK293 cells assessed as inhibition of GLP1-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGastric inhibitory polypeptide receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at mouse GIPR expressed in CHO-K1 cells assessed as inhibition of GIP-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Mouse)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at mouse GLP1R expressed in CHO-K1 cells assessed as inhibition of GLP1-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
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