Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50015064
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582404(CHEMBL5092703)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582404(CHEMBL5092703)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582405(CHEMBL5074603)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataEC50:  0.0880nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582407(CHEMBL5071417)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataEC50:  0.770nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582405(CHEMBL5074603)
Affinity DataEC50:  0.390nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataEC50:  0.0980nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataEC50:  0.380nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582407(CHEMBL5071417)
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at 3xHA tagged human CB2 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582411(CHEMBL5084325)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582411(CHEMBL5084325)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582408(CHEMBL5080279)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582412(CHEMBL5087407)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582405(CHEMBL5074603)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582400(CHEMBL5077315)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582402(CHEMBL5080450)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582408(CHEMBL5080279)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582412(CHEMBL5087407)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582409(CHEMBL5081699)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582406(CHEMBL5091754)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582407(CHEMBL5071417)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582400(CHEMBL5077315)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582400(CHEMBL5077315)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582404(CHEMBL5092703)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582408(CHEMBL5080279)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582405(CHEMBL5074603)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582407(CHEMBL5071417)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582404(CHEMBL5092703)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582405(CHEMBL5074603)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582409(CHEMBL5081699)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582404(CHEMBL5092703)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582411(CHEMBL5084325)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582407(CHEMBL5071417)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582401(CHEMBL5081770)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582409(CHEMBL5081699)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582402(CHEMBL5080450)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582402(CHEMBL5080450)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Mouse)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582412(CHEMBL5087407)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55940 from mouse CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50066712((6aR,9R,10aR)-3-(1,1-Dimethyl-heptyl)-9-hydroxymet...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by TopCount scintilla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 55 total ) | Next | Last >>
Jump to: