Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50011977
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataKd:  44nMAssay Description:Binding affinity to immobilized HDAC4 catalytic domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataKd:  3.90E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataKd: >5.00E+3nMAssay Description:Displacement of [3H]pirenzapine from human recombinant M1 receptor incubated for 1 hr by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataKd: >5.00E+3nMAssay Description:Displacement of [3H]AF-DX384 from human recombinant M2 receptor incubated for 1 hr by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataKd: >5.00E+3nMAssay Description:Displacement of [3H]4-DAMP from human recombinant M3 receptor incubated for 1 hr by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataKd: >5.00E+3nMAssay Description:Displacement of [3H]4-DAMP from human recombinant M4 receptor incubated for 1 hr by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552912(CHEMBL4760047)
Affinity DataIC50: 2nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552909(CHEMBL4754665)
Affinity DataIC50: 3nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 3nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC5 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM243178((R)-N-(1-(Azepan-1-yl)propan-2-yl)-4- (5-(trifluor...)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162839(US9056843, 130)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC7 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC9 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552909(CHEMBL4754665)
Affinity DataIC50: 10nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552912(CHEMBL4760047)
Affinity DataIC50: 10nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162840(US9056843, 131)
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC7 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC5 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 20nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552908(CHEMBL4753102)
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM243178((R)-N-(1-(Azepan-1-yl)propan-2-yl)-4- (5-(trifluor...)
Affinity DataIC50: 30nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552919(CHEMBL4747488)
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC9 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552911(CHEMBL4797931)
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 40nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552916(CHEMBL4740322)
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552918(CHEMBL3910908)
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552908(CHEMBL4753102)
Affinity DataIC50: 60nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162839(US9056843, 130)
Affinity DataIC50: 70nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM162840(US9056843, 131)
Affinity DataIC50: 70nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552919(CHEMBL4747488)
Affinity DataIC50: 70nMAssay Description:Inhibition of HDAC9 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552914(CHEMBL4764348)
Affinity DataIC50: 70nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552919(CHEMBL4747488)
Affinity DataIC50: 90nMAssay Description:Inhibition of HDAC5 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552911(CHEMBL4797931)
Affinity DataIC50: 100nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552910(CHEMBL4752150)
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552919(CHEMBL4747488)
Affinity DataIC50: 140nMAssay Description:Inhibition of HDAC7 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552916(CHEMBL4740322)
Affinity DataIC50: 180nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552913(CHEMBL4752226)
Affinity DataIC50: 230nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552919(CHEMBL4747488)
Affinity DataIC50: 250nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552917(CHEMBL4753030)
Affinity DataIC50: 280nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552917(CHEMBL4753030)
Affinity DataIC50: 310nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552910(CHEMBL4752150)
Affinity DataIC50: 380nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552914(CHEMBL4764348)
Affinity DataIC50: 600nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552918(CHEMBL3910908)
Affinity DataIC50: 730nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552923(CHEMBL4799829)
Affinity DataIC50: 890nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552913(CHEMBL4752226)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Class 2A HDAC4 in human Jurkat E6.1 cells using Boc-Lys-(TFA)-AMC as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Charles River Discovery

Curated by ChEMBL
LigandPNGBDBM50552915(CHEMBL4798111)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) using Boc-Lys(TFA) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
LigandPNGBDBM162846(US9056843, 137)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of HDAC3/NCOR2 (unknown origin) using Boc-Lys(Ac) as substrate by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
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