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Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50015599
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587744(CHEMBL5177936)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of human BuchE preincubated for 6 mins followed by substrate addition and measured upto 3 mins using acetylthiocholine iodide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587756(CHEMBL5206601)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of equine serum BuchE preincubated for 6 mins followed by substrate addition using butyrylthiocholine iodide as substrate by DTNB reagent ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587755(CHEMBL5171929)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of equine serum BuchE preincubated for 6 mins followed by substrate addition using butyrylthiocholine iodide as substrate by DTNB reagent ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587756(CHEMBL5206601)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human BuchE preincubated for 6 mins followed by substrate addition using butyrylthiocholine iodide as substrate by DTNB reagent based E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587755(CHEMBL5171929)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human BuchE preincubated for 6 mins followed by substrate addition using butyrylthiocholine iodide as substrate by DTNB reagent based E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587756(CHEMBL5206601)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human AchE preincubated for 6 mins followed by substrate addition using acetylthiocholine iodide as substrate by DTNB reagent based Ell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50510839(CHEMBL4536838)
Affinity DataIC50: 10nMAssay Description:Inhibition of equine BuChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587756(CHEMBL5206601)
Affinity DataIC50: 12nMAssay Description:Inhibition of electric eel AchE preincubated for 6 mins followed by substrate addition using acetylthiocholine iodide as substrate by DTNB reagent ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50362851(CHEMBL1940390)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate preincubated for 15 mins followed by enzyme addition and further incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587755(CHEMBL5171929)
Affinity DataIC50: 19nMAssay Description:Inhibition of human AchE preincubated for 6 mins followed by substrate addition using acetylthiocholine iodide as substrate by DTNB reagent based Ell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587744(CHEMBL5177936)
Affinity DataIC50: 20nMAssay Description:Inhibition of human AchE preincubated for 6 mins followed by substrate addition and measured upto 3 mins using acetylthiocholine iodide as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587755(CHEMBL5171929)
Affinity DataIC50: 21nMAssay Description:Inhibition of electric eel AchE preincubated for 6 mins followed by substrate addition using acetylthiocholine iodide as substrate by DTNB reagent ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50510850(CHEMBL4552675)
Affinity DataIC50: 22nMAssay Description:Inhibition of human AchE preincubated for 20 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587743(CHEMBL5199151)
Affinity DataIC50: 62nMAssay Description:Inhibition of AchE (unknown origin) using acetylcholine iodide as substrate preincubated for 10 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50510850(CHEMBL4552675)
Affinity DataIC50: 68nMAssay Description:Inhibition of human BuchE preincubated for 20 mins followed by substrate addition using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587753(CHEMBL5190569)
Affinity DataIC50: 68nMAssay Description:Inhibition of human AchE using acetylthiocholine iodide as substrate by Ellman colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587742(CHEMBL5169512)
Affinity DataIC50: 90nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587754(CHEMBL5197518)
Affinity DataIC50: 92nMAssay Description:Inhibition of human AchE using acetylthiocholine iodide as substrate by Ellman colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587743(CHEMBL5199151)
Affinity DataIC50: 107nMAssay Description:Inhibition of BuchE (unknown origin) using butylthicoline iodide as substrate preincubated for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587750(CHEMBL4087621)
Affinity DataIC50: 110nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition and measured after 5 mins using S-butyrylthiocholine iodide a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587741(CHEMBL5196661)
Affinity DataIC50: 130nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587746(CHEMBL5205151)
Affinity DataIC50: 150nMAssay Description:Inhibition of human BuchE preincubated for 30 mins followed by substrate addition using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587751(CHEMBL4096250)
Affinity DataIC50: 150nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition and measured after 5 mins using S-butyrylthiocholine iodide a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587749(CHEMBL5188267)
Affinity DataIC50: 170nMAssay Description:Inhibition of human BuchE preincubated for 30 mins followed by substrate addition using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 190nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587754(CHEMBL5197518)
Affinity DataIC50: 210nMAssay Description:Inhibition of human BuchE using butyrylthiocholine iodide as substrate by Ellman colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetBeta-secretase 1(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587754(CHEMBL5197518)
Affinity DataIC50: 210nMAssay Description:Inhibition of human BACE-1 by FRET-based fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587753(CHEMBL5190569)
Affinity DataIC50: 255nMAssay Description:Inhibition of human BuchE using butyrylthiocholine iodide as substrate by Ellman colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetBeta-secretase 1(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587753(CHEMBL5190569)
Affinity DataIC50: 255nMAssay Description:Inhibition of human BACE-1 by FRET-based fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587740(CHEMBL3819231)
Affinity DataIC50: 390nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587748(CHEMBL5194599)
Affinity DataIC50: 430nMAssay Description:Inhibition of human BuchE preincubated for 30 mins followed by substrate addition using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50195819(CHEMBL3818089)
Affinity DataIC50: 650nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587740(CHEMBL3819231)
Affinity DataIC50: 970nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition using S-butyrylthiocholine iodide as substrate by Ellman's me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587739(CHEMBL3818086)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50195819(CHEMBL3818089)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition using S-butyrylthiocholine iodide as substrate by Ellman's me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition and measured after 5 mins using S-butyrylthiocholine iodide a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of equine BuChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587739(CHEMBL3818086)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by substrate addition using S-butyrylthiocholine iodide as substrate by Ellman's me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587745(CHEMBL5200969)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as measuring amount of 4-hydroxyquinoline using kynuramine as substrate incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50515337(CHEMBL4560240)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of GluN1/GluN2B NMDA receptor (unknown origin) expressed in xenopus laevis oocytes with holding potential of -70 mV by two-electrode volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587757(CHEMBL5174092)
Affinity DataIC50: 7.03E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate incubated for 15 mins by Amplex Red reagent based fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587752(CHEMBL5187221)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human AchE preincubated for 15 mins followed by substrate addition and measured for 5 mins using acetylthiocholine iodide as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587745(CHEMBL5200969)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as measuring amount of 4-hydroxyquinoline using kynuramine as substrate incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Horse)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587745(CHEMBL5200969)
Affinity DataIC50: 8.93E+3nMAssay Description:Inhibition of equine BuChE incubated for 15 mins using using butyrylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587758(CHEMBL5184096)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins by Amplex Red reagent based fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587745(CHEMBL5200969)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of electric eel AChE incubated for 15 mins using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587757(CHEMBL5174092)
Affinity DataIC50: 2.41E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins by Amplex Red reagent based fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587747(CHEMBL5199756)
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of electric eel AchE preincubated for 30 mins followed by substrate addition using acetylthiocholine iodide as substrate by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCholinesterase(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587747(CHEMBL5199756)
Affinity DataIC50: 2.92E+4nMAssay Description:Inhibition of human BuchE preincubated for 30 mins followed by substrate addition using butyrylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Indian Institute of Technology (Banaras Hindu University)

Curated by ChEMBL
LigandPNGBDBM50587758(CHEMBL5184096)
Affinity DataIC50: 5.03E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate incubated for 15 mins by Amplex Red reagent based fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
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