Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50013183
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50563441(CHEMBL4745810)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50563442(CHEMBL4754685)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50563440(CHEMBL4784051)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50563439(CHEMBL4748649)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]-CQ transport incubated for 1.5 hrs by m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed