Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50013177
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563421(CHEMBL4745232)
Affinity DataIC50: 2.51E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563421(CHEMBL4745232)
Affinity DataIC50: 2.70E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563421(CHEMBL4745232)
Affinity DataIC50: 3.80E+3nMAssay Description:Allosteric antagonist activity at NPY5R in mouse descending colon mucosa assessed as reduction in rPP-induced ion transport by electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563421(CHEMBL4745232)
Affinity DataIC50: 3.80E+3nMAssay Description:Allosteric antagonist activity at NPY5R in mouse descending colon mucosa assessed as reduction in rPP-induced ion transport by electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563420(CHEMBL4780125)
Affinity DataIC50: 3.98E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50563420(CHEMBL4780125)
Affinity DataIC50: 4.00E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed