Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50012701
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559506(CHEMBL4756251)
Affinity DataEC50:  363nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559494(CHEMBL4759054)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559493(CHEMBL4793741)
Affinity DataEC50:  676nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559492(CHEMBL4776518)
Affinity DataEC50:  141nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50248604((3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl...)
Affinity DataEC50:  155nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559495(CHEMBL4796513)
Affinity DataEC50:  39nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559496(CHEMBL4741155)
Affinity DataEC50:  2.75E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559501(CHEMBL4752997)
Affinity DataEC50:  2.82E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559503(CHEMBL4747418)
Affinity DataEC50:  4.90E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM181239(US9139546, 26)
Affinity DataEC50:  1.66E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559505(CHEMBL4777102)
Affinity DataEC50:  372nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataEC50:  1.70E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559508(CHEMBL4749825)
Affinity DataEC50:  240nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant cannabinoid CB1 receptor expressed in HEK cells transfected with CNG assessed as decrease in cAMP level measure...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as decrease in cAMP level measure...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559493(CHEMBL4793741)
Affinity DataEC50:  1.29E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559508(CHEMBL4749825)
Affinity DataEC50:  3.47E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataEC50:  8.91E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559506(CHEMBL4756251)
Affinity DataEC50:  6.03E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559505(CHEMBL4777102)
Affinity DataEC50:  1.41E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM181239(US9139546, 26)
Affinity DataEC50: <1.00E+4nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559495(CHEMBL4796513)
Affinity DataEC50:  8.51E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559494(CHEMBL4759054)
Affinity DataEC50:  6.17E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at cannabinoid CB1 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559492(CHEMBL4776518)
Affinity DataEC50: <1.00E+4nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50248604((3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl...)
Affinity DataEC50:  155nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataEC50:  1.18E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50248604((3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559495(CHEMBL4796513)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559493(CHEMBL4793741)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559508(CHEMBL4749825)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559505(CHEMBL4777102)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559506(CHEMBL4756251)
Affinity DataKi:  233nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM181239(US9139546, 26)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559492(CHEMBL4776518)
Affinity DataKi:  447nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559494(CHEMBL4759054)
Affinity DataKi:  975nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559496(CHEMBL4741155)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559501(CHEMBL4752997)
Affinity DataKi:  1.84E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559505(CHEMBL4777102)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559502(CHEMBL4792566)
Affinity DataKi:  2.49E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559493(CHEMBL4793741)
Affinity DataKi:  3.74E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM181239(US9139546, 26)
Affinity DataKi:  4.02E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559503(CHEMBL4747418)
Affinity DataKi:  4.74E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50248604((3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl...)
Affinity DataKi:  4.78E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559491(CHEMBL4741108)
Affinity DataKi:  8.38E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559494(CHEMBL4759054)
Affinity DataKi:  9.53E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559490(CHEMBL4786835)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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