Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50035727
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  0.800nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023395((4-{3-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat brain membrane(KD)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataIC50: 16nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50367678(CHEMBL605469)
Affinity DataIC50: 430nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of photolabeling of 24 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of photolabeling of 34 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of photolabeling of 24 kDa polypeptide in adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed