Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50011495
Affinity DataKd: 243nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKd: 463nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKd: 594nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant LSD1 (158 to end residues) expressed in Escherichia coli using dimethylated H3K4 peptide as substrate by horseradish ...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of human recombinant LSD1 using ARTK(diMe)QTARKSTGGKAPRKQLA as substrate incubated for 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) cells using H3K4me2 as substrate incubated for 30 mins by horseradish pero...More data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:Inhibition of C-terminal His/FLAG-tagged human HDAC1 expressed in Sf9 insect cells using acetylated P53(379-382 residues) (RHKK(Ac)) as substrate inc...More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of LSD1/FLAG-tagged CoREST (unknown origin) expressed in HEK293F cells using diMeK4H3(1 to 21 residues) as substrate preincubated for 5 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of LSD1 (unknown origin) (157 to 852 residues) expressed in Escherichia coli BL21(DE) cells using H3K4me2 as substrate by horseradish pero...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of LSD1 (unknown origin) (157 to 852 residues) expressed in Escherichia coli BL21(DE) cells using H3K4me2 as substrate by horseradish pero...More data for this Ligand-Target Pair
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of LSD1 (unknown origin) expressed in human MGC-803 cells incubated for 5 days by DAPI staining based immunofluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...More data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of human LSD1 preincubated for 10 mins followed by H3(1-20)K4-dimethylated (K4me2) peptide substrate addition and measured after 30 mins b...More data for this Ligand-Target Pair
