Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50011989
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM429521(med.21724, Compound Gemcitabine)
Affinity DataIC50: 190nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553100(CHEMBL4800221)
Affinity DataIC50: 380nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553102(CHEMBL4764619)
Affinity DataIC50: 381nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553101(CHEMBL4796317)
Affinity DataIC50: 384nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553099(CHEMBL4746302)
Affinity DataIC50: 1.00E+3nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553098(CHEMBL4778383)
Affinity DataIC50: 1.00E+3nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50553097(CHEMBL4749693)
Affinity DataIC50: 1.00E+3nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed