Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50011988
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331042(2-(2-(((4R,8S,11S)-11-amino-8-(4-hydroxybenzyl)-6,...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553093(CHEMBL4762305)
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553092(CHEMBL4753417)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553095(CHEMBL4745618)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553096(CHEMBL4787513)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553091(CHEMBL4778960)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553090(CHEMBL4744066)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553094(CHEMBL4761376)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human IRAP expressed in HEK293T cells assessed as substrate cleavage using Leu-MCA as substrate by fluorogenic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331042(2-(2-(((4R,8S,11S)-11-amino-8-(4-hydroxybenzyl)-6,...)
Affinity DataKi:  11nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553093(CHEMBL4762305)
Affinity DataKi:  24nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553090(CHEMBL4744066)
Affinity DataKi: >100nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553094(CHEMBL4761376)
Affinity DataKi: >100nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553092(CHEMBL4753417)
Affinity DataKi:  201nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553095(CHEMBL4745618)
Affinity DataKi:  674nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553096(CHEMBL4787513)
Affinity DataKi:  887nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50553091(CHEMBL4778960)
Affinity DataKi:  1.25E+3nMAssay Description:Binding affinity to recombinant full length human IRAP expressed in HEK293T cells using Leu-MCA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed