Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50013831
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570140(CHEMBL4863321)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50077017(CHEMBL3416725)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570142(CHEMBL4878060)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50245396(CHEMBL4101200)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50245396(CHEMBL4101200)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570141(CHEMBL4875775)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of human ERAP2 assessed as hydrolysis of KSIINFEKL to SIINFEKL measured after 2 hrs by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570140(CHEMBL4863321)
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of human ERAP2 assessed as hydrolysis of KSIINFEKL to SIINFEKL measured after 2 hrs by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570143(CHEMBL4853168)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570144(CHEMBL4849358)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant ERAP2 (unknown origin) expressed in baculovirus infected Hi-5 insect cells using R-AMC as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50570140(CHEMBL4863321)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human IRAP expressed in HEK293 cells using L-AMC as substrate preincubated for 30 mins followed by substrate addition measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50077017(CHEMBL3416725)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Institut Pasteur De Lille

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 7.55E+5nMAssay Description:Inhibition of human ERAP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)