Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50012910
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK9/cyclinT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 112nMAssay Description:Inhibition of CDK4/cyclinD (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 138nMAssay Description:Inhibition of CDK1/cyclinB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 159nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 186nMAssay Description:Inhibition of CDK5/p25 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 233nMAssay Description:Inhibition of CDK2/cyclinA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 367nMAssay Description:Inhibition of CDK2/cyclinE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 399nMAssay Description:Inhibition of CDK3/cyclinE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50561527(CHEMBL4764481)
Affinity DataIC50: 555nMAssay Description:Inhibition of CDK7/cyclinH/MAT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed