Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50002563
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023004(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 180nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023001(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 200nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023002(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 540nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023016(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 560nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023017(ethyl 4-[2-(4-ethyloxycarbonylbenzyloxy)-1-(1H-1-i...)
Affinity DataIC50: 700nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023007(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.10E+3nMAssay Description:Compound was tested for inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023006(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.26E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM7962(CHEMBL537708 | 4-[2-(1H-imidazol-1-yl)ethoxy]benzo...)
Affinity DataIC50: 1.29E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023009(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.49E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023010(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.61E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023003(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.94E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023001(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 2.00E+3nMAssay Description:Compound was tested for inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023018(4-[3-Imidazol-1-yl-2-(4-methoxy-benzyloxy)-propoxy...)
Affinity DataIC50: 3.60E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023002(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 5.30E+3nMAssay Description:Compound was tested for inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023014(N-Butyl-4-[2-imidazol-1-yl-1-(4-methoxy-benzyloxym...)
Affinity DataIC50: 5.40E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023015(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 6.00E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50022999(5-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 6.20E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50022998(1-[3-(4-Methoxy-benzyloxy)-2-(4-methylsulfanyl-ben...)
Affinity DataIC50: 6.40E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023007(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 6.70E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023009(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 7.10E+3nMAssay Description:Compound was tested for inhibitory activity against human platelet microsomal TXA2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023013(3-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 7.20E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023008(1-[2-(4-Methanesulfinyl-benzyloxy)-3-(4-methoxy-be...)
Affinity DataIC50: 8.60E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023005(1-[2,3-Bis-(4-methoxy-benzyloxy)-propyl]-1H-imidaz...)
Affinity DataIC50: 9.90E+3nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023000(N-Ethyl-4-[2-imidazol-1-yl-1-(4-methoxy-benzyloxym...)
Affinity DataIC50: 1.24E+4nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023019(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.24E+4nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023011(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 2.10E+4nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023012(1-[2-(4-Methanesulfonyl-benzyloxy)-3-(4-methoxy-be...)
Affinity DataIC50: 2.49E+4nMAssay Description:Tested for inhibitory activity against intact human platelet TXA2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed