Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50013020
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562182(CHEMBL4744466)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562185(CHEMBL4746910)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562179(CHEMBL4739972)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562176(CHEMBL4778377)
Affinity DataKi:  5.10nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562184(CHEMBL4744206)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562183(CHEMBL4760742)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562181(CHEMBL4747537)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562180(CHEMBL4796195)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562186(CHEMBL4761905)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562177(CHEMBL4763056)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562179(CHEMBL4739972)
Affinity DataKi:  160nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562173(CHEMBL4778965)
Affinity DataKi:  956nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562187(CHEMBL4765186)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562178(CHEMBL4740343)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562186(CHEMBL4761905)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562185(CHEMBL4746910)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562184(CHEMBL4744206)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562183(CHEMBL4760742)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562182(CHEMBL4744466)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562181(CHEMBL4747537)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562180(CHEMBL4796195)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562178(CHEMBL4740343)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562177(CHEMBL4763056)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562176(CHEMBL4778377)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562175(CHEMBL4749663)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562174(CHEMBL4759158)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562187(CHEMBL4765186)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562175(CHEMBL4749663)
Affinity DataKi:  3.18E+3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562173(CHEMBL4778965)
Affinity DataKi:  3.19E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma intracellular receptor 2(Rat)
Guangdong Medical University

Curated by ChEMBL
LigandPNGBDBM50562174(CHEMBL4759158)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed