Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50018361
TargetCystic fibrosis transmembrane conductance regulator(Rat)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  70nMAssay Description:Potentiation of CFTR F508del mutant in rat FRT cells assessed as increase in iodide influx in presence of forskolinMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataEC50:  7.00E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50486732(CHEMBL2068831)
Affinity DataEC50:  90nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50486733(CHEMBL2068832)
Affinity DataEC50:  1.10E+3nMAssay Description:Potentiation of CFTR F508del mutant activity (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  2.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516902(CHEMBL1583913)
Affinity DataEC50:  3.80E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  3.90E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516906(CHEMBL4444246)
Affinity DataEC50:  5.00E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516908(CHEMBL4444352)
Affinity DataEC50:  4.20E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  1.40E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516902(CHEMBL1583913)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516901(CHEMBL1403454)
Affinity DataEC50:  1.50E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516906(CHEMBL4444246)
Affinity DataEC50:  3.80E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of Palermo

Curated by ChEMBL
LigandPNGBDBM50516908(CHEMBL4444352)
Affinity DataEC50:  1.10E+4nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in rat FRT cells assessed as increase in iodide influx in presence of forskolin incuba...More data for this Ligand-Target Pair
In DepthDetails
PubMed