Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50012795
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataKd: <1nMAssay Description:Binding affinity to ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataEC50:  24nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataEC50:  2nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560386(CHEMBL4743649)
Affinity DataIC50: 2nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataIC50: 3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 13nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 14nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560389(CHEMBL4744428)
Affinity DataIC50: 17nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560388(CHEMBL4753983)
Affinity DataIC50: 31nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212285(CHEMBL3891901)
Affinity DataIC50: 55nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 63nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 63nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50505941(CHEMBL4451125)
Affinity DataIC50: 100nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560387(CHEMBL4748155)
Affinity DataIC50: 130nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 200nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 251nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 270nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 631nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212282(CHEMBL3981026)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetEphrin type-A receptor 3(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetEphrin type-A receptor 3(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50212270(CHEMBL3952214)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Takeda Research In California

Curated by ChEMBL
LigandPNGBDBM50560385(CHEMBL4759397)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed