Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50011320
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3(Human)
University of Rijeka
Curated by ChEMBL
University of Rijeka
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of JAK in human PBMC assessed as inhibition of GM-CSF-induced STAT5 phosphorylation preincubated for 30 mins followed by addition IL2 stim...More data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3(Human)
University of Rijeka
Curated by ChEMBL
University of Rijeka
Curated by ChEMBL
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of JAK in human PBMC assessed as inhibition of IFNalpha-induced STAT1 phosphorylation preincubated for 30 mins followed by addition IL2 st...More data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3(Human)
University of Rijeka
Curated by ChEMBL
University of Rijeka
Curated by ChEMBL
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of JAK in human PBMC assessed as inhibition of IL2-induced STAT5 phosphorylation preincubated for 30 mins followed by addition IL2 stimula...More data for this Ligand-Target Pair
