Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012751
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM35723(N-[4-(7-Chloro-5-hydroxy-2,3,4,5-tetrahydro-benzo[...)
Affinity DataIC50: 0.00700nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559938(CHEMBL154668)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at HTR2C in human U2OS cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559937(CHEMBL4758081)
Affinity DataIC50: 459nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559937(CHEMBL4758081)
Affinity DataIC50: 1.16E+3nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProlactin-releasing peptide receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50: 4.89E+3nMAssay Description:Antagonist activity at human PRLHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50: 7.29E+3nMAssay Description:Antagonist activity at human CCR8 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in mouse C2C12 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetFollicle-stimulating hormone receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50: 8.03E+3nMAssay Description:Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50: 8.30E+3nMAssay Description:Antagonist activity at human CCR3 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCX3C chemokine receptor 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50: 8.47E+3nMAssay Description:Antagonist activity at human CX3CR1 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed