Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50007702
TargetTaste receptor type 2 member 1(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataEC50:  1.50E+5nMAssay Description:Agonist activity at TAS2R1 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 14(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at TAS2R14 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211355(US9247759, 12-6)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211364(US9247759, 12-15)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211356(US9247759, 12-7)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211358(US9247759, 12-9)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211264(US9247759, 10-12)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211353(US9247759, 12-4)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211350(US9247759, 12-1)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211270(US9247759, 10-18)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211272(US9247759, 10-20)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211263(US9247759, 10-11)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211359(US9247759, 12-10)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211261(US9247759, 10-9)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211259(US9247759, 10-7)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211273(US9247759, 10-21)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511890(CHEMBL4514970)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210974(US9247759, 4-8)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211244(US9247759, 9-1)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211305(US9247759, 10-88 | US9247759, 10-53)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210975(US9247759, 4-9)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511886(CHEMBL4452065)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211326(US9247759, 10-74)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211285(US9247759, 10-33)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211052(US9247759, 4-88)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511892(CHEMBL4469393)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211307(US9247759, 10-55)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211020(US9247759, 4-55)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211271(US9247759, 10-19)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511893(CHEMBL4567380)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511894(CHEMBL4447100)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210983(US9247759, 4-17)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210973(US9247759, compound B | US9247759, 4-7)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211021(US9247759, 4-56)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210972(US9247759, 4-6)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511888(CHEMBL4456506)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211253(US9247759, 10-1)
Affinity DataIC50: 900nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211325(US9247759, 10-73)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511896(CHEMBL4526144)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210987(US9247759, 4-21)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211306(US9247759, 10-54)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511887(CHEMBL4588973)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511891(CHEMBL4530528)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511889(CHEMBL4579065)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211011(US9247759, 4-46)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210989(US9247759, 4-24)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM210985(US9247759, 4-19)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211260(US9247759, 10-8)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetTaste receptor type 2 member 8(Human)
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511884(CHEMBL4471870)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
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