Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50010809
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM14777(CHEMBL779 | (6R,12aR)-6-(1,3-benzodioxol-5-yl)-2-m...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 86nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542291(CHEMBL4642376)
Affinity DataIC50: 110nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542297(CHEMBL4638267)
Affinity DataIC50: 260nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542295(CHEMBL4639873)
Affinity DataIC50: 330nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542277(CHEMBL4638436)
Affinity DataIC50: 610nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542292(CHEMBL4643394)
Affinity DataIC50: 630nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542293(CHEMBL4641767)
Affinity DataIC50: 790nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542294(CHEMBL4648832)
Affinity DataIC50: 970nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542289(CHEMBL4635740)
Affinity DataIC50: 970nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542275(CHEMBL4636071)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542278(CHEMBL4636060)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50131046(CHEMBL85139 | cid_65752 | rutaecarpine | 8,13-Dihy...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542290(CHEMBL4642482)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542288(CHEMBL4638725)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542276(CHEMBL4633115)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542281(CHEMBL4640216)
Affinity DataIC50: 6.17E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542282(CHEMBL4634019)
Affinity DataIC50: 9.19E+3nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542279(CHEMBL4642224)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542280(CHEMBL4635413)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542286(CHEMBL4635055)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542285(CHEMBL4639525)
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542287(CHEMBL4635751)
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50131049(11-Methoxy-8,13-dihydro-7H-indolo[2',3':3,4]pyrido...)
Affinity DataIC50: 2.21E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 3.21E+4nMAssay Description:Inhibition of PDE10 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetO43924/P16499/P18545/P35913/P51160/Q13956(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 4.38E+4nMAssay Description:Inhibition of PDE6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542283(CHEMBL4643201)
Affinity DataIC50: 4.56E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542284(CHEMBL4649889)
Affinity DataIC50: 4.73E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PDE2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PDE4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50542296(CHEMBL4641729)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PDE9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed