Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50009332
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527393(CHEMBL4446895)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527392(CHEMBL4540791)
Affinity DataIC50: 6.54E+3nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527395(CHEMBL4475137)
Affinity DataIC50: 9.82E+3nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527401(CHEMBL4542006)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527391(CHEMBL4557551)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527397(CHEMBL4566254)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527400(CHEMBL4474925)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50467448(CHEMBL4280001)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527394(CHEMBL4447706)
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527398(CHEMBL4468954)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527399(CHEMBL1092945)
Affinity DataIC50: 5.29E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527396(CHEMBL4469422)
Affinity DataIC50: 7.24E+4nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527402(CHEMBL4587427)
Affinity DataIC50: 3.84E+5nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527403(CHEMBL4450694)
Affinity DataIC50: 8.75E+5nMAssay Description:Inhibition of C-terminal 6His-tagged wild type human GYS1 using UDPG as substrate in presence of 1 mM G-6-P by 14C-glucose incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlycogen [starch] synthase, muscle(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50527393(CHEMBL4446895)
Affinity DataKi:  1.31E+3nMAssay Description:Competitive inhibition of C-terminal 6His-tagged human GYS1 using UDPG as substrate in presence of G-6-P by 14C-glucose incorporation based Michaelis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed