Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50010807
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542263(CHEMBL4638430)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542259(CHEMBL4644500)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542258(CHEMBL4634009)
Affinity DataEC50:  2nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542257(CHEMBL4640409)
Affinity DataEC50:  7nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542256(CHEMBL4648027)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542255(CHEMBL4636321)
Affinity DataEC50:  12nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542254(CHEMBL4633978)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542253(CHEMBL4635414)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542252(CHEMBL4644352)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542251(CHEMBL4647011)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542250(CHEMBL4638599)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542260(CHEMBL4644742)
Affinity DataEC50:  20nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542250(CHEMBL4638599)
Affinity DataEC50:  14nMAssay Description:Agonist activity at D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataEC50:  27nMAssay Description:Agonist activity at D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50073444(2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}[1,2...)
Affinity DataEC50:  785nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM194780(US9206167, 1 | brexpiprazole | 7-(4-(4-(1-benzothi...)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542267(CHEMBL4649106)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542266(CHEMBL4633397)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542265(CHEMBL4636764)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542264(CHEMBL4635890)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataEC50:  9.70nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542262(CHEMBL4648979)
Affinity DataEC50:  5.90nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin) by calcium-dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542263(CHEMBL4638430)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542266(CHEMBL4633397)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542267(CHEMBL4649106)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542258(CHEMBL4634009)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542250(CHEMBL4638599)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM25870(CITALOPRAM HYDROBROMIDE | [3H]Escitalopram | Escit...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at SERT receptor (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542258(CHEMBL4634009)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542265(CHEMBL4636764)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542250(CHEMBL4638599)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542252(CHEMBL4644352)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542251(CHEMBL4647011)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542253(CHEMBL4635414)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542252(CHEMBL4644352)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542252(CHEMBL4644352)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542250(CHEMBL4638599)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542252(CHEMBL4644352)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542265(CHEMBL4636764)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542260(CHEMBL4644742)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542251(CHEMBL4647011)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542253(CHEMBL4635414)
Affinity DataIC50: 63nMAssay Description:Antagonist activity at D2 receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542266(CHEMBL4633397)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542259(CHEMBL4644500)
Affinity DataIC50: 85nMAssay Description:Antagonist activity at 5HT2A receptor (unknown origin) by HTRF cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50542261(CHEMBL4644391)
Affinity DataIC50: 88nMAssay Description:Antagonist activity at alpha-1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
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