Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50011810
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  0.00630nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551315(CHEMBL4762529)
Affinity DataKi:  0.0125nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  0.0136nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  0.0220nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  0.0240nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551309(CHEMBL4758369)
Affinity DataKi:  0.0325nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  0.0333nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  0.0435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  0.177nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  0.214nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551312(CHEMBL4761619)
Affinity DataKi:  0.218nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551317(CHEMBL4764372)
Affinity DataKi:  0.252nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551312(CHEMBL4761619)
Affinity DataKi:  0.257nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551308(CHEMBL4758814)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  0.321nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551318(CHEMBL4787652)
Affinity DataKi:  0.326nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551310(CHEMBL4752367)
Affinity DataKi:  0.435nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551308(CHEMBL4758814)
Affinity DataKi:  0.531nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551317(CHEMBL4764372)
Affinity DataKi:  0.682nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  0.796nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551311(CHEMBL4746512)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551316(CHEMBL4776706)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551307(CHEMBL4754079)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551314(CHEMBL4751305)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551315(CHEMBL4762529)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551319(CHEMBL4753839)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551313(CHEMBL4745764)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551309(CHEMBL4758369)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551310(CHEMBL4752367)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551318(CHEMBL4787652)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]HS665 from KOR in guinea pig brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551315(CHEMBL4762529)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551312(CHEMBL4761619)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551308(CHEMBL4758814)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551317(CHEMBL4764372)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551310(CHEMBL4752367)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551309(CHEMBL4758369)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Szeged

Curated by ChEMBL
LigandPNGBDBM50551318(CHEMBL4787652)
Affinity DataKi:  3.91E+3nMAssay Description:Displacement of [3H]Ile5'6-deltorphin II from DOR in Wistar rat brain membranes measured after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed