Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50007119
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506506(CHEMBL4465833)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506504(CHEMBL4460663)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506505(CHEMBL4460376)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506498(CHEMBL4581886)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506501(CHEMBL4563019)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506500(CHEMBL4471611)
Affinity DataIC50: 1nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506499(CHEMBL4463265)
Affinity DataIC50: 2nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187287(US9169240, 27)
Affinity DataIC50: 3nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506505(CHEMBL4460376)
Affinity DataIC50: 4nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506506(CHEMBL4465833)
Affinity DataIC50: 4nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506499(CHEMBL4463265)
Affinity DataIC50: 5nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187290(US9169240, 30)
Affinity DataIC50: 5nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506500(CHEMBL4471611)
Affinity DataIC50: 9nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187289(US9169240, 29)
Affinity DataIC50: 10nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506497(CHEMBL4446812)
Affinity DataIC50: 10nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187310(US9169240, 49)
Affinity DataIC50: 10nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187290(US9169240, 30)
Affinity DataIC50: 10nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187289(US9169240, 29)
Affinity DataIC50: 10nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506503(CHEMBL4475891)
Affinity DataIC50: 20nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506502(CHEMBL4575712)
Affinity DataIC50: 20nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187287(US9169240, 27)
Affinity DataIC50: 20nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506500(CHEMBL4471611)
Affinity DataIC50: 20nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506498(CHEMBL4581886)
Affinity DataIC50: 20nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506501(CHEMBL4563019)
Affinity DataIC50: 20nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506504(CHEMBL4460663)
Affinity DataIC50: 20nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506497(CHEMBL4446812)
Affinity DataIC50: 20nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187286(US9169240, 26)
Affinity DataIC50: 30nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506502(CHEMBL4575712)
Affinity DataIC50: 30nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506503(CHEMBL4475891)
Affinity DataIC50: 30nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187310(US9169240, 49)
Affinity DataIC50: 30nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506498(CHEMBL4581886)
Affinity DataIC50: 40nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506503(CHEMBL4475891)
Affinity DataIC50: 40nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506501(CHEMBL4563019)
Affinity DataIC50: 40nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506506(CHEMBL4465833)
Affinity DataIC50: 50nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHepatic triacylglycerol lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187285(US9169240, 25)
Affinity DataIC50: 60nMAssay Description:Inhibition of human HL expressed in human COS7 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506499(CHEMBL4463265)
Affinity DataIC50: 60nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506504(CHEMBL4460663)
Affinity DataIC50: 60nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187285(US9169240, 25)
Affinity DataIC50: 90nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506497(CHEMBL4446812)
Affinity DataIC50: 100nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506499(CHEMBL4463265)
Affinity DataIC50: 100nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50506504(CHEMBL4460663)
Affinity DataIC50: 200nMAssay Description:Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506505(CHEMBL4460376)
Affinity DataIC50: 200nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50506505(CHEMBL4460376)
Affinity DataIC50: 200nMAssay Description:Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187286(US9169240, 26)
Affinity DataIC50: 200nMAssay Description:Inhibition of EL in human HT1080 cells using A10070 as substrate preincubated for 20 min followed by DMPG vesicle doped substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50506498(CHEMBL4581886)
Affinity DataIC50: 200nMAssay Description:Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50506506(CHEMBL4465833)
Affinity DataIC50: 200nMAssay Description:Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187285(US9169240, 25)
Affinity DataIC50: 200nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187289(US9169240, 29)
Affinity DataIC50: 200nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187289(US9169240, 29)
Affinity DataIC50: 200nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetEndothelial lipase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM187290(US9169240, 30)
Affinity DataIC50: 400nMAssay Description:Inhibition of EL in human HT1080 cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of human serum by LC/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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