Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50010500
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539626(CHEMBL4642708)
Affinity DataIC50: 4nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539625(CHEMBL4640664)
Affinity DataIC50: 4nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539636(CHEMBL4641234)
Affinity DataIC50: 4nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539627(CHEMBL4646285)
Affinity DataIC50: 6nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM86612(Benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one, 1...)
Affinity DataIC50: 7nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539635(CHEMBL4645836)
Affinity DataIC50: 7nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539628(CHEMBL4648763)
Affinity DataIC50: 11nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539637(CHEMBL4640785)
Affinity DataIC50: 13nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539621(CHEMBL4640316)
Affinity DataIC50: 16nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539641(CHEMBL4635845)
Affinity DataIC50: 18nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539616(CHEMBL4640243)
Affinity DataIC50: 26nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539639(CHEMBL4644425)
Affinity DataIC50: 26nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539643(CHEMBL4647099)
Affinity DataIC50: 28nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539632(CHEMBL4639490)
Affinity DataIC50: 29nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539631(CHEMBL4639091)
Affinity DataIC50: 37nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539629(CHEMBL4647423)
Affinity DataIC50: 37nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539630(CHEMBL4637921)
Affinity DataIC50: 41nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50337126(US9266890, IV-2 | CHEMBL1672987 | Scaffold, B19 | ...)
Affinity DataIC50: 44nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539642(CHEMBL4645704)
Affinity DataIC50: 50nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539633(CHEMBL4646592)
Affinity DataIC50: 62nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539624(CHEMBL4648368)
Affinity DataIC50: 63nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539634(CHEMBL4644218)
Affinity DataIC50: 66nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539614(CHEMBL4649556)
Affinity DataIC50: 73nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539622(CHEMBL4637720)
Affinity DataIC50: 88nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539640(CHEMBL4633821)
Affinity DataIC50: 91nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539623(CHEMBL4634637)
Affinity DataIC50: 97nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539618(CHEMBL4642494)
Affinity DataIC50: 101nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539644(CHEMBL4648786)
Affinity DataIC50: 140nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539615(CHEMBL4633699)
Affinity DataIC50: 217nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539613(CHEMBL4636937)
Affinity DataIC50: 223nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539638(CHEMBL4644196)
Affinity DataIC50: 254nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539617(CHEMBL4645012)
Affinity DataIC50: 308nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539612(CHEMBL4644397)
Affinity DataIC50: 363nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539619(CHEMBL4635766)
Affinity DataIC50: 723nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50337127(US9266890, IV-1 | 2-(2-methoxy-4-(4-methylpiperazi...)
Affinity DataIC50: 959nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539611(CHEMBL4646229)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50539620(CHEMBL4642279)
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of tracer 236 binding to recombinant human GST-tagged TNK2 catalytic domain (110 to 476 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed