Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50008527
TargetTubulin beta chain(Pig)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50520178(CHEMBL4468642)
Affinity DataKd:  2.66E+3nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetTubulin beta chain(Pig)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50014846(7alphaH-colchicine | (S)-N-(5,6,7,9-tetrahydro-1,2...)
Affinity DataKd:  1.13E+4nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetTubulin beta chain(Pig)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50520178(CHEMBL4468642)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured at 30 secs interval for 65 mins by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed