Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50009516
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529555(CHEMBL4524997)
Affinity DataKd:  1.71E+4nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529557(CHEMBL4588022)
Affinity DataKd:  1.81E+4nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  6.10E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466619(CHEMBL4290656)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  113nMAssay Description:Binding affinity to human MLLT1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529558(CHEMBL4456056)
Affinity DataKd:  5.50E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529559(CHEMBL4444396)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 260nMAssay Description:Inhibition of human MLLT1 by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529558(CHEMBL4456056)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466619(CHEMBL4290656)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529559(CHEMBL4444396)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529557(CHEMBL4588022)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50529555(CHEMBL4524997)
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)