Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50009701
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531293(CHEMBL4471671)
Affinity DataIC50: 417nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531293(CHEMBL4471671)
Affinity DataIC50: 417nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531299(CHEMBL4454608)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531299(CHEMBL4454608)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531300(CHEMBL4455491)
Affinity DataIC50: 1.48E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531300(CHEMBL4455491)
Affinity DataIC50: 1.48E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531305(CHEMBL4453937)
Affinity DataIC50: 1.86E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531305(CHEMBL4453937)
Affinity DataIC50: 1.86E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531298(CHEMBL4592514)
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531298(CHEMBL4592514)
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531296(CHEMBL4451522)
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531296(CHEMBL4451522)
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human A1AR expressed in CHO-K1 cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  0.302nMAssay Description:Antagonist activity at A2AR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  0.302nMAssay Description:Antagonist activity at A2AR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531293(CHEMBL4471671)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531293(CHEMBL4471671)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531299(CHEMBL4454608)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531299(CHEMBL4454608)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531300(CHEMBL4455491)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531300(CHEMBL4455491)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531298(CHEMBL4592514)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531298(CHEMBL4592514)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531305(CHEMBL4453937)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531305(CHEMBL4453937)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531307(CHEMBL4471931)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531307(CHEMBL4471931)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531296(CHEMBL4451522)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531296(CHEMBL4451522)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  2.04E+3nMAssay Description:Antagonist activity at A1AR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  2.04E+3nMAssay Description:Antagonist activity at A1AR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531309(CHEMBL4532681)
Affinity DataKi:  3.02E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531309(CHEMBL4532681)
Affinity DataKi:  3.02E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531308(CHEMBL1731061)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531308(CHEMBL1731061)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531295(CHEMBL4471221)
Affinity DataKi:  6.92E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531295(CHEMBL4471221)
Affinity DataKi:  6.92E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531306(CHEMBL4445436)
Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531306(CHEMBL4445436)
Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531294(CHEMBL4528096)
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531294(CHEMBL4528096)
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531304(CHEMBL4583555)
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531304(CHEMBL4583555)
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531310(CHEMBL4513678)
Affinity DataKi:  1.86E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531310(CHEMBL4513678)
Affinity DataKi:  1.86E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531297(CHEMBL4525388)
Affinity DataKi:  1.95E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531297(CHEMBL4525388)
Affinity DataKi:  1.95E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531302(CHEMBL1397091)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531302(CHEMBL1397091)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531301(CHEMBL4449779)
Affinity DataKi:  2.57E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531301(CHEMBL4449779)
Affinity DataKi:  2.57E+4nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cells incubated for 50 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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