Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50007961
TargetGuanine nucleotide binding protein, alpha q polypeptide(Chinese hamster)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514449(CHEMBL4171381)
Affinity DataIC50: 33nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGuanine nucleotide binding protein, alpha q polypeptide(Chinese hamster)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 95nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM114291(8-(3,4,5-trihydroxy-6-oxoxanthen-9-yl)naphthalene-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514448(CHEMBL4469620)
Affinity DataIC50: 200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50246208(cid_274122 | CHEMBL487046 | 2-(3,4,5-trihydroxy-6-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514450(CHEMBL4443974)
Affinity DataIC50: 250nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50444748(Aminoquinuride)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM97335(SMR001566795 | MLS002702986 | 7-amino-1,2,3,10-tet...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514451(CHEMBL1967787)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of G-protein beta1gamma2 (unknown origin) by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed