Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50009697
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 98nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 98nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 400nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 400nMAssay Description:Inhibition of human SIRT2 (25-389 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 400nMAssay Description:Inhibition of human SIRT2 (25-389 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 400nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531283(CHEMBL4452438)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531283(CHEMBL4452438)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of SIRT1 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of SIRT1 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.98E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.98E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531288(CHEMBL4553883)
Affinity DataIC50: 6.77E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531288(CHEMBL4553883)
Affinity DataIC50: 6.77E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531287(CHEMBL4454236)
Affinity DataIC50: 8.57E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531287(CHEMBL4454236)
Affinity DataIC50: 8.57E+3nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531284(CHEMBL4456147)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531284(CHEMBL4456147)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531289(CHEMBL4443075)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531289(CHEMBL4443075)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM29040(cambinol)
Affinity DataIC50: 3.88E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM29040(cambinol)
Affinity DataIC50: 3.88E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531285(CHEMBL4581121)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.98E+4nMAssay Description:Inhibition of SIRT3 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 4.98E+4nMAssay Description:Inhibition of SIRT3 (unknown origin) using fluorogenic substrate assessed as deacetylase activity incubated for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM29040(cambinol)
Affinity DataIC50: 4.99E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) assessed as increase in alpha-tubulin acetylation after 2 hrs by alpha-tubulin acetyl-K40 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM29040(cambinol)
Affinity DataIC50: 4.99E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) assessed as increase in alpha-tubulin acetylation after 2 hrs by alpha-tubulin acetyl-K40 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) assessed as increase in alpha-tubulin acetylation after 2 hrs by alpha-tubulin acetyl-K40 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531286(CHEMBL4568936)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) assessed as increase in alpha-tubulin acetylation after 2 hrs by alpha-tubulin acetyl-K40 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human SIRT1 (133-747 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531283(CHEMBL4452438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50531283(CHEMBL4452438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human SIRT1 (133-747 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human SIRT3 (101-399 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human SIRT3 (101-399 aa) expressed in Escherichia coli BL21 using ZMAL (Z-Lys(Acetyl)-AMC) as substrate incubated for 4 hrs by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50148800(CHEMBL3770486)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed