Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50010452
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539037(CHEMBL4645684)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539042(CHEMBL4646737)
Affinity DataKd:  20nMAssay Description:Binding affinity to LPA1 receptor (unknown origin) by cell-based backscattering interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataKd:  5.60nMAssay Description:Binding affinity to LPA1 receptor (unknown origin) by cell-based backscattering interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539046(CHEMBL4636192)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539045(CHEMBL4648653)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539044(CHEMBL4648374)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539043(CHEMBL4648051)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539042(CHEMBL4646737)
Affinity DataEC50:  240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539041(CHEMBL4643694)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539040(CHEMBL4637403)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539039(CHEMBL4637898)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539038(CHEMBL4644847)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50:  221nMAssay Description:Agonist activity at LPA1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539036(CHEMBL4636453)
Affinity DataEC50:  500nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539035(CHEMBL4642688)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539034(CHEMBL4642952)
Affinity DataEC50:  240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539033(CHEMBL4632820)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539032(CHEMBL4633208)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539031(CHEMBL4643262)
Affinity DataEC50:  450nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539030(CHEMBL4647245)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50539029(CHEMBL4646443)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at recombinant human full-length LPA1 receptor expressed in dhfr- deficient CHO cells assessed as increase in intracellular calcium ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at LPA2 (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed