Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50011762
TargetProtein disulfide-isomerase A3(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A6(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A6(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetThioredoxin domain-containing protein 5(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A6(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A3(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A3(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A4(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50: 3.31E+4nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A4(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: 6.16E+4nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein disulfide-isomerase A4(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetThioredoxin domain-containing protein 5(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetThioredoxin domain-containing protein 5(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed