Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50012641
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558959(CHEMBL4740594)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558957(CHEMBL4755128)
Affinity DataKd:  3.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558967(CHEMBL4759563)
Affinity DataKd:  8.5nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558956(CHEMBL4743733)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human MetAP1 expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558959(CHEMBL4740594)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558962(CHEMBL4783117)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558960(CHEMBL4758588)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558961(CHEMBL4741746)
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558958(CHEMBL4743353)
Affinity DataIC50: 9.87E+4nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558954(CHEMBL4749821)
Affinity DataIC50: 1.04E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558966(CHEMBL4752621)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558963(CHEMBL4795438)
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558953(CHEMBL4745980)
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558964(CHEMBL4777085)
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558951(CHEMBL4759464)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558955(CHEMBL4784882)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558965(CHEMBL4785449)
Affinity DataIC50: 1.43E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558952(CHEMBL4764436)
Affinity DataIC50: 1.75E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558957(CHEMBL4755128)
Affinity DataIC50: 2.17E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
University of Hyderabad

Curated by ChEMBL
LigandPNGBDBM50558956(CHEMBL4743733)
Affinity DataIC50: 2.84E+5nMAssay Description:Inhibition of human MetAP1 expressed in Escherichia coli BL21 (DE3) using L-methionine-4-methyl-coumary1-7-amide as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed