Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50006935
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50148603(CHEMBL3770724)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504782(CHEMBL4567799)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504783(CHEMBL4582177)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504780(CHEMBL4466089)
Affinity DataIC50: 4.11E+6nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504781(CHEMBL4448567)
Affinity DataIC50: 6.88E+6nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50353587(CHEMBL12543)
Affinity DataIC50: 2.66E+6nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504784(CHEMBL4570065)
Affinity DataIC50: 4.81E+6nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50504785(CHEMBL4538721)
Affinity DataIC50: 2.12E+6nMAssay Description:Inhibition of GST-tagged BRD4 BD1 (49 to 170 residues) (unknown origin) using streptavidin-D2 biotinylated tetra-acetylated histone H4 peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed